| Nombre | MARIO FERNANDEZ ZERTUCHE |
|---|---|
| Área | BIOLOGÍA Y QUÍMICA |
| Campo | QUÍMICA |
| Disciplina | QUÍMICA GENERAL |
| Especialidad | QUIMICA ORGANICA MEDICINAL |
| CVU | 15480 |
| Institución |
SIN INSTITUCIÓN
|
|---|---|
| Dependencia | NO APLICA |
| Entidad | NO APLICA |
| Nivel | 2 |
| Vigencia | Inicio: 01/01/2022 |
| Fin: 31/12/2036 | |
| Categoría: | EXTENSION 15 AÑOS |
Publicaciones ORCID
- 2025
- Computer‐Aided Drug Design of (R)‐Baclofen Isoxazole and Tetrazole Derivatives: Searching for Novel GABAB Receptor Agonists ChemistrySelect
- 2024
- Design and synthesis of 3,5-disubstituted isoxazoles by Cu-mediated 1,3-dipolar cycloaddition and their in silico evaluation as potential GABAB receptor modulators Tetrahedron
- 2021
- Preclinical safety evaluation of amphotericin A21: A novel antifungal Basic & Clinical Pharmacology & Toxicology
- 2020
- 1,4‐Disubstituted‐1,2,3‐triazole GABA Analogues: Synthesis, In Vitro Evaluation, Quantum QSAR and Molecular Docking against Pseudomonas fluorescens GABA‐AT ChemistrySelect
- 2019
- In silico structure‐based design of GABAB receptor agonists using a combination of docking and QSAR Chemical Biology & Drug Design
- 2018
- QSAR and Molecular Docking Studies of the Inhibitory Activity of Novel Heterocyclic GABA Analogues over GABA-AT Molecules
- Novel-Substituted Heterocyclic GABA Analogues. Enzymatic Activity against the GABA-AT Enzyme from Pseudomonas fluorescens and In Silico Molecular Modeling Molecules
- 2016
- An Amphotericin B Derivative Equally Potent to Amphotericin B and with Increased Safety PlosOne
- Multigram Scale Synthesis of A21, A New Antibiotic Equally Effective and Less Toxic than Amphotericin B Org. Process Res. Dev. 2016, 20, 1529−1532
